| 生物活性 |
Lumateperone-d4 (ITI-007-d4) is deuterium labeled Lumateperone. Lumateperone (ITI-007) is an orally active 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone has anticancer activity and can also be used for the study of schizophrenia and bipolar depression.
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| 分子式 |
C24H24D4FN3O
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| 分子量 |
397.52
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| CAS号 |
2102683-55-4
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| 运输条件 |
Room temperature in continental US; may vary elsewhere.
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| 储存方式 |
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Data Sheet
