Farletuzumab ecteribulin
(Synonyms:(MORAb-202))
目录号 : KM36787
CAS No. : 2407465-18-1
纯度 : 98%
Farletuzumab ecteribulin (MORAb-202) 是一种抗体-活性分子偶联物 (ADC),由人源化抗人叶酸受体 α (FRA) 抗体 Farletuzumab 通过还原的链间二硫键与 Mal-PEG2-Val-Cit-PAB-eribulin 偶联而成。Farletuzumab ecteribulin 的活性分子抗体比为 4.0。Farletuzumab ecteribulin 在体外对 FRA 阳性细胞具有高度细胞毒性。Farletuzumab ecteribulin 具有有效的抗肿瘤活性。
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| 生物活性 |
Farletuzumab ecteribulin (MORAb-202) is an antibody-drug conjugate (ADC), consisting of the humanized anti-human folate receptor alpha (FRA) antibody Farletuzumab conjugated via reduced interchain disulfide bonds to Mal-PEG2-Val-Cit-PAB-eribulin. Farletuzumab ecteribulin has a agent-to-antibody ratio of 4.0. Farletuzumab ecteribulin is highly cytotoxic to FRA-positive cells in vitro. Farletuzumab ecteribulin has potent antitumor activity.
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| 分子量 |
149000 (average)
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| CAS号 |
2407465-18-1
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| 运输条件 |
Shipping with dry ice.
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| 储存方式 |
| Powder |
-20°C |
3 years |
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4°C |
2 years |
| In solvent |
-80°C |
6 months |
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-20°C |
1 month |
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