Pantoprazole-d4
(Synonyms:BY1023-d4)
目录号 : KM37245
CAS No. : 934294-71-0
Pantoprazole-d4 (BY1023-d4) 是氘代标记的 Pantoprazole. Pantoprazole (BY1023) 是一种具有口服活性的,有效质子泵 (proton pump) 抑制剂 (PPI)。Pantoprazole 是一种取代的苯并咪唑,是一种有效的 H+/K+-ATPase 抑制剂,IC50 为 6.8 μM。Pantoprazo 可以改善 pH 值稳定性,并具有抗分泌,抗溃疡的作用。Pantoprazo 联合阿霉素 (Doxorubicin) 可显着增加肿瘤生长延迟。
Other Forms of Rapamycin:
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| 生物活性 |
Pantoprazole-d4 (BY1023-d4) is deuterium labeled Pantoprazole. Pantoprazole (BY10232) is an orally active and potent proton pump inhibitor (PPI). Pantoprazole, a substituted benzimidazole, is a potent H+/K+-ATPase inhibitor with an IC50 of 6.8 μM. Pantoprazole improves pH stability and has anti-secretory, anti-ulcer activities. Pantoprazole significantly increased tumor growth delay combined with Doxorubicin .
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| 分子式 |
C16H11D4F2N3O4S
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| 分子量 |
387.39
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| CAS号 |
934294-71-0
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| 运输条件 |
Room temperature in continental US; may vary elsewhere.
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| 储存方式 |
| Powder |
-20°C |
3 years |
| |
4°C |
2 years |
| In solvent |
-80°C |
6 months |
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-20°C |
1 month |
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