Labetalol hydrochloride-d5
(Synonyms:盐酸拉贝洛尔-d5)
目录号 : KM38454
CAS No. : 2713514-78-2
Labetalol hydrochloride-d5 (AH-5158 hydrochloride-d5) 是氘代标记的 Labetalol hydrochloride 。Labetalol (AH5158) hydrochloride 是一种口服有效的、选择性 α1- 和非选择性 β-肾上腺素能受体 (adrenergic receptor) 竞争性拮抗剂。Labetalol hydrochloride 是一种抗高血压活性分子,可部分透过血脑屏障,且对心输出量影响较小。Labetalol hydrochloride 可用于心血管疾病的研究,如妊娠期高血压。
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| 生物活性 |
Labetalol hydrochloride-d5 (AH-5158 hydrochloride-d5) is deuterium labeled Labetalol hydrochloride . Labetalol (AH5158) hydrochloride is an orally available, selective α1-adrenergic recepto and non-selective β-adrenergic receptor competitive antagonist. Labetalol hydrochloride is an antihypertensive molecule that partially crosses the blood-brain barrier and has little effect on cardiac output. Labetalol hydrochloride can be used in the study of cardiovascular diseases, such as hypertension during pregnancy.
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| 分子式 |
C19H20D5ClN2O3
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| 分子量 |
369.9
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| CAS号 |
2713514-78-2
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| 运输条件 |
Room temperature in continental US; may vary elsewhere.
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| 储存方式 |
| Powder |
-20°C |
3 years |
| |
4°C |
2 years |
| In solvent |
-80°C |
6 months |
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-20°C |
1 month |
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