DP-C-4 是一种基于 Cereblon 的双 PROTAC,用于同时降解 EGFR 和 PARP。
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DP-C-4 is a Cereblon-based dual PROTAC for simultaneous degradation of EGFR and PARP.
DP-C-4 (1-50 μM; 24 hours) has degradation effects on EGFR and PARP simultaneously in a dose-dependent manner in SW1990 cells.
Western Blot Analysis
Room temperature in continental US; may vary elsewhere.
-80°C, stored under nitrogen
DMSO : 12 mg/mL (8.27 mM; Need ultrasonic)
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纯度: 98%
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