Certepetide - CAS:2580154-02-3

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Certepetide (Synonyms:NRP-1激活剂;CEND-1; iRGD; LSTA1)

目录号 : KM24936 CAS No. : 2580154-02-3 纯度 : 98%

Data Sheet 产品使用指南

Certepetide (CEND-1) is a bifunctional cyclic peptide (a.k.a. iRGD). Certepetide is a tumor-penetrating enhancer via RGD motif interaction with alphav-integrins and via activating NRP-1, and transforms the solid tumor microenvironment into a temporary drug conduit. Certepetide accumulates in tumors, and is used in the research of pancreatic cancer and other solid tumors.

规格	价格	是否有货
1mg		In-stock
5mg		In-stock
10mg		In-stock
50mg	询价	In-stock
100mg	询价	In-stock

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生物活性

体内研究

CEND-1 (iRGD) can regulate the solid tumor microenvironment, enhance the delivery and therapeutic index of co administered anticancer drugs.

CEND-1 can enhance the specific penetration of anti-cancer drugs into tumors rather than normal tissues, while also having the potential to reduce dosage and alleviate side effects.

CEND-1 (intravenous injection) will increase the effectiveness of Evans blue when administered in combination by about three times.

分子式

C₃₇H₆₀N₁₄O₁₄S₂

分子量

989.09

CAS号

2580154-02-3

中文名称

NRP-1激活剂

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

-20°C,Sealed storage, away from moisture and light, under nitrogen

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light, under nitrogen)

溶解性数据

In Vitro:

H2O : ≥ 50 mg/mL (50.55 mM)

DMSO : 2.33 mg/mL (2.36 mM; Need ultrasonic)

* "≥" means soluble, but saturation unknown.

配制储备液

浓度溶剂体积质量	1 mg	5 mg	10 mg

1 mM	1.0110 mL	5.0552 mL	10.1103 mL
5 mM	0.2022 mL	1.0110 mL	2.0221 mL
10 mM	0.1011 mL	0.5055 mL	1.0110 mL

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light, under nitrogen)。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。

纯度： 98%