AG-041R - CAS:159883-95-1

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AG-041R

目录号 : KCM11761 CAS No. : 159883-95-1 纯度 : ≥98%

Data Sheet 产品使用指南

The peptide hormone gastrin acts through G protein-coupled cholecystokinin-2 (CCK) receptors to regulate cell proliferation, differentiation, apoptosis, and gene expression of gastrointestinal cells and exerts trophic effects on a number of gastric cancer cell lines. AG-041R is a potent gastrin/CCK receptor antagonist that exhibits selective binding for CCK compared to CCK AG-041R inhibits gastrin-evoked secretion of pancreastatin (IC = 2.2 nM) as well as gastrin-induced histamine release and cell growth of Mastomys ECL carcinoid tumor cells. AG-041R (1 µM) exhibits synergistic inhibitory effects on the cell viability of human gastric cancer cells when administered in combination with the selective COX-2 inhibitor NS-398 at 10 µM.

规格	价格	是否有货	数量
1mg		In-stock
5mg		In-stock
10mg		In-stock
50mg		In-stock

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AG-041R In-stock

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生物活性

AG-041R is a potent and selective CCK2 Receptor/Gastrin antagonist. AG-041R inhibits gastrin-evoked secretion of pancreastatin with an IC₅₀ of 2.2 nM. AG-041R inhibits cell growth of Mastomys ECL carcinoid tumor cells.

分子式

C₃₁H₃₆N₄O₅

分子量

544.7

CAS号

159883-95-1

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Powder	-20°C	3 years
In solvent	-80°C	6 months
	-20°C	1 month

纯度： ≥98%

Data Sheet

产品使用指南

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

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Other Forms of Rapamycin:

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